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【简答题】
β-内酰胺类抗生素的构效关系与哪项不符 A. β-内酰胺环是抗菌作用的必要结构,β-内酰胺环并合六元的氢化噻嗪环可显著提高抗菌活性 B. 6-氨基或7-氨基的酰化侧链影响抗菌强度,抗菌谱,耐青霉素酶及耐酸性 C. 侧链中引入吸电子基团将增强对酸的稳定性 D.侧链中引入体积较大基团可增强对青霉素酶的稳定性 E.头孢菌素类的3-位取代基的改变,主要影响化合物的药物动力学特性
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